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Search Results for " nicotinic receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T28531 Facinicline hydrochloride RG3487 5-HT Receptor , AChR
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM). Facinicline hydrochloride improves cognition and sensorimot...
T60080 TMPH 2,2,6,6-Tetramethylpiperidin-4-yl heptanoate AChR
TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.
T1039 Choline chloride Biocolina,Biocoline,Hepacholine AChR
Choline chloride (Biocoline) is a basic constituent of lecithin that is found in many plants and animal organs. It is important as a precursor of acetylcholine, as a methyl donor in various metabolic processes, and in li...
T2198 Arecoline hydrobromide Arecoline HBr,Arecoline bromide AChR
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.
T22448 Tropisetron Tropisetronum,Tropisteron,ICS 205-930 5-HT Receptor , AChR
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.
T23146 PHA 568487 free base PHA 568487 AChR
The quinuclidine PHA 568487 free base is an agonist of the alpha 7 nicotinic acetylcholine receptor that was designed to mitigate the bioactivation associated with the core scaffold and subsequently remove associated lia...
T22016 A-582941 dihydrochloride A 582941 5-HT Receptor , AChR
A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial
T8040 Cholesterol myristate Cholesteryl myristate,Cholesteryl tetradecanoate Others , Potassium Channel , GABA Receptor , Endogenous Metabolite , AChR
Cholesterol Myristate (Cholesteryl Myristate) is a natural steroid found in traditional Chinese medicine that interacts with various ion channels, including the GABAA receptor, nicotinic acetylcholine receptor, and the i...
T2227 Hemicholinium 3 Hemicholinium-3,Hemicholine Others , AChE
Hemicholinium 3 is a potent and selective choline uptake blocker.
T2663 GTS-21 dihydrochloride GTS 21 dihydrochloride,DMXB-A,DMBX-anabaseine 5-HT Receptor , AChR
GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.
T2141 Mecamylamine hydrochloride Inversine,Mevasin AChR
Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
T12525 Pozanicline dihydrochloride ABT-089 dihydrochloride AChR
Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)
T3023 Catharanthine sulfate AChR
Catharanthine inhibits nicotinic receptor-mediated diaphragm contractions.
T0268 Lobeline hydrochloride α-Lobeline hydrochloride,L-Lobeline hydrochloride AChR
Lobeline hydrochloride (α-Lobeline hydrochloride) is a nicotinic receptor agonist, acting as an effective antagonist at both α4β2 and α3β2 neuronal nicotinic receptor subtypes.
T12820 S16961 S169611 AChR
S16961 (S169611) is an agonist of nicotinic receptor.
T2782 Catharanthine (+)-3, 4-Didehydrocoronaridine,(+)-3,4-Didehydrocoronaridine Calcium Channel , AChR
Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
T37818 BPiDDB N,N'-Dodecylbis-Picolinium Bromide AChR
bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.
T12738L1 Rivanicline 2HCl Rivanicline 2HCl(15585-43-0 Free base) AChR
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.
T12017 Methyllycaconitine citrate MLA AChR
Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.
T10914 Cyclodrine hydrochloride AChR
Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of neurologically related diseases.

Compounds

Facinicline hydrochloride
T28531
Synonym: RG3487
Target: 5-HT Receptor, AChR
TMPH
T60080
Synonym: 2,2,6,6-Tetramethylpiperidin-4-yl heptanoate
Target: AChR
Choline chloride
T1039
Synonym: Biocolina,Biocoline,Hepacholine
Target: AChR
Arecoline hydrobromide
T2198
Synonym: Arecoline HBr,Arecoline bromide
Target: AChR
Tropisetron
T22448
Synonym: Tropisetronum,Tropisteron,ICS 205-930
Target: 5-HT Receptor, AChR
PHA 568487 free base
T23146
Synonym: PHA 568487
Target: AChR
A-582941 dihydrochloride
T22016
Synonym: A 582941
Target: 5-HT Receptor, AChR
Cholesterol myristate
T8040
Synonym: Cholesteryl myristate,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
Hemicholinium 3
T2227
Synonym: Hemicholinium-3,Hemicholine
Target: Others, AChE
GTS-21 dihydrochloride
T2663
Synonym: GTS 21 dihydrochloride,DMXB-A,DMBX-anabaseine
Target: 5-HT Receptor, AChR
Mecamylamine hydrochloride
T2141
Synonym: Inversine,Mevasin
Target: AChR
Pozanicline dihydrochloride
T12525
Synonym: ABT-089 dihydrochloride
Target: AChR
Catharanthine sulfate
T3023
Synonym:
Target: AChR
Lobeline hydrochloride
T0268
Synonym: α-Lobeline hydrochloride,L-Lobeline hydrochloride
Target: AChR
S16961
T12820
Synonym: S169611
Target: AChR
Catharanthine
T2782
Synonym: (+)-3, 4-Didehydrocoronaridine,(+)-3,4-Didehydrocoronaridine
Target: Calcium Channel, AChR
bPiDDB
T37818
Synonym: N,N'-Dodecylbis-Picolinium Bromide
Target: AChR
Rivanicline 2HCl
T12738L1
Synonym: Rivanicline 2HCl(15585-43-0 Free base)
Target: AChR
Methyllycaconitine citrate
T12017
Synonym: MLA
Target: AChR
Cyclodrine hydrochloride
T10914
Synonym:
Target: AChR
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TargetMol